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Reaction Details
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TargetAdenosine receptor A1
LigandBDBM50452271
Substrate/Competitorn/a
Meas. Tech.ChEBML_29298
Ki 20000±n/a nM
Citation Taylor, MDMoos, WHHamilton, HWSzotek, DSPatt, WCBadger, EWBristol, JABruns, RFHeffner, TGMertz, TE Ribose-modified adenosine analogues as adenosine receptor agonists. J Med Chem29:346-53 (1986) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Adenosine receptor A1
Name:Adenosine receptor
Synonyms:ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptors A1
Type:Protein
Mol. Mass.:36704.13
Organism:Rattus norvegicus (rat)
Description:n/a
Residue:326
Sequence:
MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVT
QRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCQPKPPIDEDLPEEKAED
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50452271
NameBDBM50452271
Synonyms:CHEMBL2111777
TypeSmall organic molecule
Emp. Form.C19H23N5O4
Mol. Mass.385.417
SMILESC[C@H](Cc1ccccc1)Nc1ncnc2n(cnc12)[C@@H]1O[C@@H](CO)[C@@H](O)[C@H]1O |r|
Structure
n/a