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Target
Adenosine receptor A1
Ligand
BDBM50008387
Substrate
n/a
Meas. Tech.
ChEBML_28960
Ki
1.5±n/a nM
Citation
 van Galen, PJ; Nissen, P; van Wijngaarden, I; IJzerman, AP; Soudijn, W 1H-imidazo[4,5-c]quinolin-4-amines: novel non-xanthine adenosine antagonists. J Med Chem 34:1202-6 (1991) [PubMed]  Article 
Target
Name:
Adenosine receptor A1
Synonyms:
AA1R_BOVIN | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | ADORA1 | Adenosine A1 receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
36602.99
Organism:
BOVINE
Description:
ADENOSINE 0 BOVINE::P28190
Residue:
326
Sequence:
MPPSISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGALVIPLAILINIGPRTYFHTCLKVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVTPRRAVVAITGCWILSFVVGLTPMFGWNNLSAVERDWLANGSVGEPVIECQFEKVISMEYMVYFNFFVWVLPPLLLMVLIYMEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALILFLFALSWLPLHILNCITLFCPSCHMPRILIYIAIFLSHGNSAMNPIVYAFRIQKFRVTFLKIWNDHFRCQPAPPVDEDAPAERPDD
  
Inhibitor
Name:
BDBM50008387
Synonyms:
CHEMBL19768 | Cyclopentyl-(2-phenyl-1H-imidazo[4,5-c]quinolin-4-yl)-amine | Cyclopentyl-(2-phenyl-1H-imidazo[4,5-c]quinolin-4-yl)-amine;HCl
Type:
Small organic molecule
Emp. Form.:
C21H20N4
Mol. Mass.:
328.4103
SMILES:
C1CCC(C1)Nc1nc2ccccc2c2nc([nH]c12)-c1ccccc1
Structure:
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