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Target
Delta-type opioid receptor
Ligand
BDBM50453048
Substrate
n/a
Meas. Tech.
ChEMBL_145892 (CHEMBL754258)
IC50
27500±n/a nM
Citation
Hruby, VJ; Toth, G; Gehrig, CA; Kao, LF; Knapp, R; Lui, GK; Yamamura, HI; Kramer, TH; Davis, P; Burks, TF Topographically designed analogues of [D-Pen,D-Pen5]enkephalin. J Med Chem 34:1823-30 (1991) [PubMed] Article
More Info.:
Target
Name:
Delta-type opioid receptor
Synonyms:
DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40577.25
Organism:
MOUSE
Description:
P32300
Residue:
372
Sequence:
MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVCAVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAALHLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTACTPSDGPGGGAAA