Reaction Details Report a problem with these data
Target
P2Y purinoceptor 1
Ligand
BDBM50369452
Substrate
n/a
Meas. Tech.
ChEMBL_147712 (CHEMBL759182)
EC50
10±n/a nM
Citation
 Fischer, B; Chulkin, A; Boyer, JL; Harden, KT; Gendron, FP; Beaudoin, AR; Chapal, J; Hillaire-Buys, D; Petit, P 2-thioether 5'-O-(1-thiotriphosphate)adenosine derivatives as new insulin secretagogues acting through P2Y-Receptors. J Med Chem 42:3636-46 (1999) [PubMed]  Article 
Target
Name:
P2Y purinoceptor 1
Synonyms:
P2RY1 | P2RY1_MELGA
Type:
n/a
Mol. Mass.:
41199.64
Organism:
Meleagris gallopavo
Description:
n/a
Residue:
362
Sequence:
MTEALISAALNGTQPELLAGGWAAGNASTKCSLTKTGFQFYYLPTVYILVFITGFLGNSVAIWMFVFHMRPWSGISVYMFNLALADFLYVLTLPALIFYYFNKTDWIFGDVMCKLQRFIFHVNLYGSILFLTCISVHRYTGVVHPLKSLGRLKKKNAVYVSSLVWALVVAVIAPILFYSGTGVRRNKTITCYDTTADEYLRSYFVYSMCTTVFMFCIPFIVILGCYGLIVKALIYKDLDNSPLRRKSIYLVIIVLTVFAVSYLPFHVMKTLNLRARLDFQTPQMCAFNDKVYATYQVTRGLASLNSCVDPILYFLAGDTFRRRLSRATRKSSRRSEPNVQSKSEEMTLNILTEYKQNGDTSL
  
Inhibitor
Name:
BDBM50369452
Synonyms:
CHEMBL611285
Type:
Small organic molecule
Emp. Form.:
C16H28N5O13P3S
Mol. Mass.:
623.406
SMILES:
CCCCCCSc1nc(N)c2ncn(C3O[C@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]3O)c2n1 |r|
Structure:
Search PDB for entries with ligand similarity: