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Target
P2X purinoceptor 5
Ligand
BDBM50368125
Substrate
n/a
Meas. Tech.
ChEMBL_147417 (CHEMBL750991)
EC50
18000±n/a nM
Citation
Jacobson, KA; Jarvis, MF; Williams, M Purine and pyrimidine (P2) receptors as drug targets. J Med Chem 45:4057-93 (2002) [PubMed] Article
More Info.:
Target
Name:
P2X purinoceptor 5
Synonyms:
ATP receptor | P2RX5_RAT | P2X5 | P2rx5 | Purinergic receptor
Type:
PROTEIN
Mol. Mass.:
51486.52
Organism:
Rattus norvegicus
Description:
ChEMBL_147417
Residue:
455
Sequence:
MGQAAWKGFVLSLFDYKTAKFVVAKSKKVGLLYRVLQLIILLYLLIWVFLIKKSYQDIDTSLQSAVVTKVKGVAYTNTTMLGERLWDVADFVIPSQGENVFFVVTNLIVTPNQRQGICAEREGIPDGECSEDDDCHAGESVVAGHGLKTGRCLRVGNSTRGTCEIFAWCPVETKSMPTDPLLKDAESFTISIKNFIRFPKFNFSKANVLETDNKHFLKTCHFSSTNLYCPIFRLGSIVRWAGADFQDIALKGGVIGIYIEWDCDLDKAASKCNPHYYFNRLDNKHTHSISSGYNFRFARYYRDPNGVEFRDLMKAYGIRFDVIVNGKAGKFSIIPTVINIGSGLALMGAGAFFCDLVLIYLIRKSEFYRDKKFEKVRGQKEDANVEVEANEMEQERPEDEPLERVRQDEQSQELAQSGRKQNSNCQVLLEPARFGLRENAIVNVKQSQILHPVKT