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TargetMu-type opioid receptor
LigandBDBM50204457
Substrate/Competitorn/a
Meas. Tech.ChEMBL_438282
Ki 4.8±n/a nM
Citation Peng, XKnapp, BIBidlack, JMNeumeyer, JL High-affinity carbamate analogues of morphinan at opioid receptors. Bioorg Med Chem Lett17:1508-11 (2007) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOP | MOR-1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | hMOP | mu-type opioid receptor isoform MOR-1
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:44789.51
Organism:Homo sapiens (Human)
Description:P35372
Residue:400
Sequence:
MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCP
PTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALAT
STLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDF
RTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFI
FAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHI
YVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNI
EQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
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  Blast E-value cutoff:
BDBM50204457
n/a
NameBDBM50204457
Synonyms:CHEMBL241823 | MCL-431
TypeSmall organic molecule
Emp. Form.C20H28N2O2
Mol. Mass.328.4485
SMILESCCNC(=O)Oc1ccc2CC3C4CCCCC4(CCN3C)c2c1 |TLB:21:20:9.22.10:12,23:22:12:20.18.19|
Structure
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