Reaction Details Report a problem with these data
Target
Nuclear receptor subfamily 4 group A member 2
Ligand
BDBM50371205
Substrate
n/a
Meas. Tech.
ChEMBL_453027 (CHEMBL902174)
EC50
31.9±n/a nM
Citation
Hintermann, S; Chiesi, M; von Krosigk, U; Mathé, D; Felber, R; Hengerer, B Identification of a series of highly potent activators of the Nurr1 signaling pathway. Bioorg Med Chem Lett 17:193-6 (2006) [PubMed] Article
More Info.:
Target
Name:
Nuclear receptor subfamily 4 group A member 2
Synonyms:
NOT | NR4A2 | NR4A2_HUMAN | NURR1 | TINUR
Type:
PROTEIN
Mol. Mass.:
66603.77
Organism:
Homo sapiens (Human)
Description:
ChEMBL_453027
Residue:
598
Sequence:
MPCVQAQYGSSPQGASPASQSYSYHSSGEYSSDFLTPEFVKFSMDLTNTEITATTSLPSFSTFMDNYSTGYDVKPPCLYQMPLSGQQSSIKVEDIQMHNYQQHSHLPPQSEEMMPHSGSVYYKPSSPPTPTTPGFQVQHSPMWDDPGSLHNFHQNYVATTHMIEQRKTPVSRLSLFSFKQSPPGTPVSSCQMRFDGPLHVPMNPEPAGSHHVVDGQTFAVPNPIRKPASMGFPGLQIGHASQLLDTQVPSPPSRGSPSNEGLCAVCGDNAACQHYGVRTCEGCKGFFKRTVQKNAKYVCLANKNCPVDKRRRNRCQYCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKSPQEPSPPSPPVSLISALVRAHVDSNPAMTSLDYSRFQANPDYQMSGDDTQHIQQFYDLLTGSMEIIRGWAEKIPGFADLPKADQDLLFESAFLELFVLRLAYRSNPVEGKLIFCNGVVLHRLQCVRGFGEWIDSIVEFSSNLQNMNIDISAFSCIAALAMVTERHGLKEPKRVEELQNKIVNCLKDHVTFNNGGLNRPNYLSKLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPAIIDKLFLDTLPF