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Target
P2Y purinoceptor 2
Ligand
BDBM50378128
Substrate
n/a
Meas. Tech.
ChEMBL_587770 (CHEMBL1040421)
IC50
264000±n/a nM
Citation
 Sauer, R; El-Tayeb, A; Kaulich, M; Müller, CE Synthesis of uracil nucleotide analogs with a modified, acyclic ribose moiety as P2Y(2) receptor antagonists. Bioorg Med Chem 17:5071-9 (2009) [PubMed]  Article 
Target
Name:
P2Y purinoceptor 2
Synonyms:
ATP receptor | P2RY2_MOUSE | P2U purinoceptor 1 | P2U1 | P2Y purinoceptor 2 | P2Y2 | P2ru1 | P2ry2 | Purinergic receptor | Purinergic receptor P2Y2
Type:
PROTEIN
Mol. Mass.:
42202.78
Organism:
Mus musculus
Description:
ChEMBL_587770
Residue:
373
Sequence:
MAADLEPWNSTINGTWEGDELGYKCRFNEDFKYVLLPVSYGVVCVLGLCLNVVALYIFLCRLKTWNASTTYMFHLAVSDSLYAASLPLLVYYYARGDHWPFSTVLCKLVRFLFYTNLYCSILFLTCISVHRCLGVLRPLHSLRWGRARYARRVAAVVWVLVLACQAPVLYFVTTSVRGTRITCHDTSARELFSHFVAYSSVMLGLLFAVPFSVILVCYVLMARRLLKPAYGTTGGLPRAKRKSVRTIALVLAVFALCFLPFHVTRTLYYSFRSLDLSCHTLNAINMAYKITRPLASANSCLDPVLYFLAGQRLVRFARDAKPPTEPTPSPQARRKLGLHRPNRTVRKDLSVSSDDSRRTESTPAGSETKDIRL
  
Inhibitor
Name:
BDBM50378128
Synonyms:
CHEMBL575653
Type:
Small organic molecule
Emp. Form.:
C8H15N2O13P3
Mol. Mass.:
440.1316
SMILES:
OP(O)(=O)OP(O)(=O)OP(O)(=O)OCCCOCn1ccc(=O)[nH]c1=O
Structure:
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