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Target
Isoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)
Ligand
BDBM50330500
Substrate
n/a
Meas. Tech.
ChEMBL_684948 (CHEMBL1286363)
IC50
96000±n/a nM
Citation
Kireev, D; Wigle, TJ; Norris-Drouin, J; Herold, JM; Janzen, WP; Frye, SV Identification of non-peptide malignant brain tumor (MBT) repeat antagonists by virtual screening of commercially available compounds. J Med Chem 53:7625-31 (2010) [PubMed] Article
More Info.:
Target
Name:
Isoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)
Synonyms:
H-l(3)mbt | H-l(3)mbt protein | KIAA0681 | L(3)mbt protein homolog | L(3)mbt-like | L3MBT | L3MBTL | L3MBTL1 | LMBL1_HUMAN | Lethal(3)malignant brain tumor-like protein 1 | Lethal(3)malignant brain tumor-like protein 1 (4) | Lethal(3)malignant brain tumor-like protein 1 (L3MBTL1)
Type:
Protein
Mol. Mass.:
83871.06
Organism:
Homo sapiens (Human)
Description:
Q9Y468-4
Residue:
752
Sequence:
MRRREGHGTDSEMGQGPVRESQSSDPPALQFRISEYKPLNMAGVEQPPSPELRQEGVTEYEDGGAPAGDGEAGPQQAEDHPQNPPEDPNQDPPEDDSTCQCQACGPHQAAGPDLGSSNDGCPQLFQERSVIVENSSGSTSASELLKPMKKRKRREYQSPSEEESEPEAMEKQEEGKDPEGQPTASTPESEEWSSSQPATGEKKECWSWESYLEEQKAITAPVSLFQDSQAVTHNKNGFKLGMKLEGIDPQHPSMYFILTVAEVCGYRLRLHFDGYSECHDFWVNANSPDIHPAGWFEKTGHKLQPPKGYKEEEFSWSQYLRSTRAQAAPKHLFVSQSHSPPPLGFQVGMKLEAVDRMNPSLVCVASVTDVVDSRFLVHFDNWDDTYDYWCDPSSPYIHPVGWCQKQGKPLTPPQDYPDPDNFCWEKYLEETGASAVPTWAFKVRPPHSFLVNMKLEAVDRRNPALIRVASVEDVEDHRIKIHFDGWSHGYDFWIDADHPDIHPAGWCSKTGHPLQPPLGPREPSSASPGGCPPLSYRSLPHTRTSKYSFHHRKCPTPGCDGSGHVTGKFTAHHCLSGCPLAERNQSRLKAELSDSEASARKKNLSGFSPRKKPRHHGRIGRPPKYRKIPQEDFQTLTPDVVHQSLFMSALSAHPDRSLSVCWEQHCKLLPGVAGISASTVAKWTIDEVFGFVQTLTGCEDQARLFKDEMIDGEAFLLLTQADIVKIMSVKLGPALKIYNAILMFKNADDTLK