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Target
Lysophosphatidic acid receptor 5
Ligand
BDBM50388091
Substrate
n/a
Meas. Tech.
ChEMBL_830366 (CHEMBL2061000)
IC50
800±n/a nM
Citation
Kozian, DH; Evers, A; Florian, P; Wonerow, P; Joho, S; Nazare, M Selective non-lipid modulator of LPA5 activity in human platelets. Bioorg Med Chem Lett 22:5239-43 (2012) [PubMed] Article
More Info.:
Target
Name:
Lysophosphatidic acid receptor 5
Synonyms:
GPR92 | GPR93 | LPAR5 | LPAR5_HUMAN | Lysophosphatidic acid receptor 5 | Lysophosphatidic acid receptor 5 (LPA5)
Type:
Enzyme
Mol. Mass.:
41372.36
Organism:
Homo sapiens (Human)
Description:
Q9H1C0
Residue:
372
Sequence:
MLANSSSTNSSVLPCPDYRPTHRLHLVVYSLVLAAGLPLNALALWVFLRALRVHSVVSVYMCNLAASDLLFTLSLPVRLSYYALHHWPFPDLLCQTTGAIFQMNMYGSCIFLMLINVDRYAAIVHPLRLRHLRRPRVARLLCLGVWALILVFAVPAARVHRPSRCRYRDLEVRLCFESFSDELWKGRLLPLVLLAEALGFLLPLAAVVYSSGRVFWTLARPDATQSQRRRKTVRLLLANLVIFLLCFVPYNSTLAVYGLLRSKLVAASVPARDRVRGVLMVMVLLAGANCVLDPLVYYFSAEGFRNTLRGLGTPHRARTSATNGTRAALAQSERSAVTTDATRPDAASQGLLRPSDSHSLSSFTQCPQDSAL