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Target
Solute carrier family 15 member 2
Ligand
BDBM50016695
Substrate
n/a
Meas. Tech.
ChEMBL_835961 (CHEMBL2077099)
Ki
6000±n/a nM
Citation
 Ramamoorthy, S; Liu, W; Ma, YY; Yang-Feng, TL; Ganapathy, V; Leibach, FH Proton/peptide cotransporter (PEPT 2) from human kidney: functional characterization and chromosomal localization. Biochim Biophys Acta 1240:1-4 (1996) [PubMed]  Article 
Target
Name:
Solute carrier family 15 member 2
Synonyms:
Kidney H(+)/peptide cotransporter | Oligopeptide transporter, kidney isoform | PEPT2 | Peptide transporter 2 | S15A2_HUMAN | SLC15A2
Type:
PROTEIN
Mol. Mass.:
81795.62
Organism:
Homo sapiens (Human)
Description:
ChEMBL_762551
Residue:
729
Sequence:
MNPFQKNESKETLFSPVSIEEVPPRPPSPPKKPSPTICGSNYPLSIAFIVVNEFCERFSYYGMKAVLILYFLYFLHWNEDTSTSIYHAFSSLCYFTPILGAAIADSWLGKFKTIIYLSLVYVLGHVIKSLGALPILGGQVVHTVLSLIGLSLIALGTGGIKPCVAAFGGDQFEEKHAEERTRYFSVFYLSINAGSLISTFITPMLRGDVQCFGEDCYALAFGVPGLLMVIALVVFAMGSKIYNKPPPEGNIVAQVFKCIWFAISNRFKNRSGDIPKRQHWLDWAAEKYPKQLIMDVKALTRVLFLYIPLPMFWALLDQQGSRWTLQAIRMNRNLGFFVLQPDQMQVLNPLLVLIFIPLFDFVIYRLVSKCGINFSSLRKMAVGMILACLAFAVAAAVEIKINEMAPAQPGPQEVFLQVLNLADDEVKVTVVGNENNSLLIESIKSFQKTPHYSKLHLKTKSQDFHFHLKYHNLSLYTEHSVQEKNWYSLVIREDGNSISSMMVKDTESRTTNGMTTVRFVNTLHKDVNISLSTDTSLNVGEDYGVSAYRTVQRGEYPAVHCRTEDKNFSLNLGLLDFGAAYLFVITNNTNQGLQAWKIEDIPANKMSIAWQLPQYALVTAGEVMFSVTGLEFSYSQAPSSMKSVLQAAWLLTIAVGNIIVLVVAQFSGLVQWAEFILFSCLLLVICLIFSIMGYYYVPVKTEDMRGPADKHIPHIQGNMIKLETKKTKL
  
Inhibitor
Name:
BDBM50016695
Synonyms:
(2S)-2-{[(2S)-2-aminopropanoyl]amino}propanoic acid | (S)-2-((S)-2-Amino-propionylamino)-propionic acid | Ala-Ala | CHEMBL17697
Type:
Small organic molecule
Emp. Form.:
C6H12N2O3
Mol. Mass.:
160.1711
SMILES:
C[C@H](N)C(=O)N[C@@H](C)C(O)=O
Structure:
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