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Target
Urotensin-2
Ligand
BDBM50414770
Substrate
n/a
Meas. Tech.
ChEMBL_588520 (CHEMBL1041260)
EC50
1096.48±n/a nM
Citation
 Lehmann, F; Currier, EA; Clemons, B; Hansen, LK; Olsson, R; Hacksell, U; Luthman, K Novel and potent small-molecule urotensin II receptor agonists. Bioorg Med Chem 17:4657-65 (2009) [PubMed]  Article 
Target
Name:
Urotensin-2
Synonyms:
UTS2 | UTS2_HUMAN
Type:
PROTEIN
Mol. Mass.:
14297.49
Organism:
Homo sapiens (Human)
Description:
ChEMBL_643307
Residue:
124
Sequence:
MYKLASCCLLFIGFLNPLLSLPLLDSREISFQLSAPHEDARLTPEELERASLLQILPEMLGAERGDILRKADSSTNIFNPRGNLRKFQDFSGQDPNILLSHLLARIWKPYKKRETPDCFWKYCV
  
Inhibitor
Name:
BDBM50414770
Synonyms:
CHEMBL574726
Type:
Small organic molecule
Emp. Form.:
C28H27ClN2O
Mol. Mass.:
442.98
SMILES:
CN(C)CCC(NC(=O)c1cccc(c1)-c1ccc(Cl)cc1)c1ccc2ccccc2c1
Structure:
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