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Target
Lysophosphatidic acid receptor 5
Ligand
BDBM50430006
Substrate
n/a
Meas. Tech.
ChEMBL_946256 (CHEMBL2344994)
EC50
6.1±n/a nM
Citation
 Jiang, G; Inoue, A; Aoki, J; Prestwich, GD Phosphorothioate analogs of sn-2 radyl lysophosphatidic acid (LPA): metabolically stabilized LPA receptor agonists. Bioorg Med Chem Lett 23:1865-9 (2013) [PubMed]  Article 
Target
Name:
Lysophosphatidic acid receptor 5
Synonyms:
GPR92 | GPR93 | LPAR5 | LPAR5_HUMAN | Lysophosphatidic acid receptor 5 | Lysophosphatidic acid receptor 5 (LPA5)
Type:
Enzyme
Mol. Mass.:
41372.36
Organism:
Homo sapiens (Human)
Description:
Q9H1C0
Residue:
372
Sequence:
MLANSSSTNSSVLPCPDYRPTHRLHLVVYSLVLAAGLPLNALALWVFLRALRVHSVVSVYMCNLAASDLLFTLSLPVRLSYYALHHWPFPDLLCQTTGAIFQMNMYGSCIFLMLINVDRYAAIVHPLRLRHLRRPRVARLLCLGVWALILVFAVPAARVHRPSRCRYRDLEVRLCFESFSDELWKGRLLPLVLLAEALGFLLPLAAVVYSSGRVFWTLARPDATQSQRRRKTVRLLLANLVIFLLCFVPYNSTLAVYGLLRSKLVAASVPARDRVRGVLMVMVLLAGANCVLDPLVYYFSAEGFRNTLRGLGTPHRARTSATNGTRAALAQSERSAVTTDATRPDAASQGLLRPSDSHSLSSFTQCPQDSAL
  
Inhibitor
Name:
BDBM50430006
Synonyms:
CHEMBL2335048
Type:
Small organic molecule
Emp. Form.:
C22H47O5PS
Mol. Mass.:
454.644
SMILES:
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(O)=S)OC |r|
Structure:
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