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Target
PHD finger protein 23
Ligand
BDBM50440608
Substrate
n/a
Meas. Tech.
ChEMBL_983401 (CHEMBL2429071)
IC50
>10000±n/a nM
Citation
 James, LI; Korboukh, VK; Krichevsky, L; Baughman, BM; Herold, JM; Norris, JL; Jin, J; Kireev, DB; Janzen, WP; Arrowsmith, CH; Frye, SV Small-molecule ligands of methyl-lysine binding proteins: optimization of selectivity for L3MBTL3. J Med Chem 56:7358-71 (2013) [PubMed]  Article 
Target
Name:
PHD finger protein 23
Synonyms:
PDH-containing protein JUNE-1 | PHD finger protein 23 | PHD finger protein 23 (PHF23) | PHF23 | PHF23_HUMAN
Type:
Protein
Mol. Mass.:
43813.67
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
403
Sequence:
MLEAMAEPSPEDPPPTLKPETQPPEKRRRTIEDFNKFCSFVLAYAGYIPPSKEESDWPASGSSSPLRGESAADSDGWDSAPSDLRTIQTFVKKAKSSKRRAAQAGPTQPGPPRSTFSRLQAPDSATLLEKMKLKDSLFDLDGPKVASPLSPTSLTHTSRPPAALTPVPLSQGDLSHPPRKKDRKNRKLGPGAGAGFGVLRRPRPTPGDGEKRSRIKKSKKRKLKKAERGDRLPPPGPPQAPPSDTDSEEEEEEEEEEEEEEMATVVGGEAPVPVLPTPPEAPRPPATVHPEGVPPADSESKEVGSTETSQDGDASSSEGEMRVMDEDIMVESGDDSWDLITCYCRKPFAGRPMIECSLCGTWIHLSCAKIKKTNVPDFFYCQKCKELRPEARRLGGPPKSGEP
  
Inhibitor
Name:
BDBM50440608
Synonyms:
CHEMBL2426374
Type:
Small organic molecule
Emp. Form.:
C29H36N4O2
Mol. Mass.:
472.6217
SMILES:
CCN1Cc2ccc(NC(=O)c3ccc(cc3)C(=O)N3CC4CCC(C3)C4N3CCCC3)cc2C1 |TLB:17:19:26:22.23|
Structure:
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