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TargetChromobox protein homolog 7 (CBX7)
LigandBDBM50440606
Substrate/Competitorn/a
Meas. Tech.ChEMBL_983405
IC50>10000±n/a nM
Citation James, LIKorboukh, VKKrichevsky, LBaughman, BMHerold, JMNorris, JLJin, JKireev, DBJanzen, WPArrowsmith, CHFrye, SV Small-molecule ligands of methyl-lysine binding proteins: optimization of selectivity for L3MBTL3. J Med Chem56:7358-71 (2013) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Chromobox protein homolog 7 (CBX7)
Name:Chromobox protein homolog 7
Synonyms:CBX7 | Chromobox protein homolog 7
Type:Protein
Mol. Mass.:28351.76
Organism:Homo sapiens (Human)
Description:n/a
Residue:251
Sequence:
MELSAIGEQVFAVESIRKKRVRKGKVEYLVKWKGWPPKYSTWEPEEHILDPRLVMAYEEK
EERDRASGYRKRGPKPKRLLLQRLYSMDLRSSHKAKGKEKLCFSLTCPLGSGSPEGVVKA
GAPELVDKGPLVPTLPFPLRKPRKAHKYLRLSRKKFPPRGPNLESHSHRRELFLQEPPAP
DVLQAAGEWEPAAQPPEEEADADLAEGPPPWTPALPSSEVTVTDITANSITVTFREAQAA
EGFFRDRSGKF
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  Blast E-value cutoff:
BDBM50440606
NameBDBM50440606
Synonyms:CHEMBL2426376
TypeSmall organic molecule
Emp. Form.C33H39N5O2
Mol. Mass.537.6951
SMILESCCN1Cc2ccc(NC(=O)c3ccc(cc3Nc3ccccc3)C(=O)N3CCC(CC3)C3CCCN3)cc2C1
Structure
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n/a