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Target
Cathepsin B
Ligand
BDBM50320734
Substrate
n/a
Meas. Tech.
ChEMBL_1337273 (CHEMBL3240887)
Ki
1900±n/a nM
Citation
 Raghav, N; Singh, M Acyl hydrazides and triazoles as novel inhibitors of mammalian cathepsin B and cathepsin H. Eur J Med Chem 77:231-42 (2014) [PubMed]  Article 
Target
Name:
Cathepsin B
Synonyms:
n/a
Type:
Protein
Mol. Mass.:
36777.57
Organism:
Capra hircus (Goat)
Description:
n/a
Residue:
335
Sequence:
MWQLLATLSCLLVLTSARSSLHFPPLSDEMVNYVNKQNTTWKAGHNFYNVDLSYVKKLCGAILGGPKLPQRDAFAADMVLPDSFDAREQWPNCPTIKEIRDQGSCGSCWAFGAVEAISDRICIHSKGRVNVEVSAEDMLTCCGSECGDGCNGGFPSGAWNFWTKKGLVSGGLYDSHVGCRPYSIPPCEHHVNGSRPPCTGEGDTPKCSKICEPGYSPSYKDDKHFGCSSYSVSSNEKEIMAEIYKNGPVEGAFSVYSDFLLYKSGVYQHVSGEMMGGHAIRILGWGVENDTPYWLVGNSWNTDWGDKGFFKILRGQDHCGIESEIVAGMPCTHQY
  
Inhibitor
Name:
BDBM50320734
Synonyms:
4-Hydroxy-benzoic acid hydrazide | 4-hydroxybenzohydrazide | CHEMBL124267
Type:
Small organic molecule
Emp. Form.:
C7H8N2O2
Mol. Mass.:
152.1506
SMILES:
NNC(=O)c1ccc(O)cc1
Structure:
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