Reaction Details Report a problem with these data
Target
Adenylate kinase 2, mitochondrial
Ligand
BDBM50010315
Substrate
n/a
Meas. Tech.
ChEMBL_1340550 (CHEMBL3254974)
Ki
320000±n/a nM
Citation
Hampton, A; Picker, D Design of species- or isozyme-specific enzyme inhibitors. 3. Species and isozymic differences between mammalian and bacterial adenylate kinases in substituent tolerance in an enzyme-substrate complex. J Med Chem 22:1529-32 (1980) [PubMed] Article
More Info.:
Target
Name:
Adenylate kinase 2, mitochondrial
Synonyms:
2.7.4.3 | AK 2 | ATP-AMP transphosphorylase 2 | ATP:AMP phosphotransferase | Adenylate kinase 2 | Adenylate kinase 2, mitochondrial | Adenylate monophosphate kinase | Ak2 | KAD2_RAT
Type:
n/a
Mol. Mass.:
26380.21
Organism:
Rattus norvegicus
Description:
n/a
Residue:
239
Sequence:
MAPNALAPEPEHPEGIRAVLLGPPGAGKGTQAPKLAENFCVCHLATGDMLRAMVASGSELGKKLKATMDAGKLVSDEMVVELIEKNLETPSCKNGFLLDGFPRTVKQAEMLDDLMDKRKEKLDSVIEFSIQDSLLIRRITGRLIHPKSGRSYHEEFNPPKEAMKDDITGEPLIRRSDDNEKALKTRLEAYHTQTTPLVEYYRKRGIHCAIDASQTPDVVFASILAAFSKATCKDLVMFV