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TargetSomatostatin receptor type 3
LigandBDBM50021091
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1365873
Ki 30±n/a nM
Citation Li, DWu, ZYu, YBall, RGGuo, LSherer, EHe, SHong, QLai, ZQi, HTruong, QYang, DXChicchi, GGTsao, KLTrusca, DTrujillo, MPachanski, MEiermann, GJHoward, ADZhou, YPZhang, BBNargund, RPHagmann, WK Diamine Derivatives as Novel Small-Molecule, Potent, and Subtype-Selective Somatostatin SST3 Receptor Agonists. ACS Med Chem Lett5:690-5 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Somatostatin receptor type 3
Name:Somatostatin receptor type 3
Synonyms:SOMATOSTATIN SST3 | SS-3-R | SS3-R | SS3R | SSR-28 | SSTR3 | Somatostatin receptor type 3 (SSTR3)
Type:Protein
Mol. Mass.:45855.97
Organism:Homo sapiens (Human)
Description:P32745
Residue:418
Sequence:
MDMLHPSSVSTTSEPENASSAWPPDATLGNVSAGPSPAGLAVSGVLIPLVYLVVCVVGLL
GNSLVIYVVLRHTASPSVTNVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLVM
AVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVVV
FSGVPRGMSTCHMQWPEPAAAWRAGFIIYTAALGFFGPLLVICLCYLLIVVKVRSAGRRV
WAPSCQRRRRSERRVTRMVVAVVALFVLCWMPFYVLNIVNVVCPLPEEPAFFGLYFLVVA
LPYANSCANPILYGFLSYRFKQGFRRVLLRPSRRVRSQEPTVGPPEKTEEEDEEEEDGEE
SREGGKGKEMNGRVSQITQPGTSGQERPPSRVASKEQQLLPQEASTGEKSSTMRISYL
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50021091
NameBDBM50021091
Synonyms:CHEMBL3287635
TypeSmall organic molecule
Emp. Form.C21H21F2N3O
Mol. Mass.369.4077
SMILESFc1ccc(cc1F)C(=O)N[C@@H]1CCC[C@H]1NCc1c[nH]c2ccccc12 |r|
Structure
n/a