Target
Cytosol aminopeptidase [33-68,L62W]
Ligand
BDBM50025099
Substrate
n/a
Meas. Tech.
ChEMBL_1442056 (CHEMBL3373424)
Ki
108±n/a nM
Citation
 Vassiliou, SWeglarz-Tomczak, EBerlicki, LPawelczak, MNocek, BMulligan, RJoachimiak, AMucha, A Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases. J Med Chem 57:8140-51 (2014) [PubMed]  Article 
Target
Name:
Cytosol aminopeptidase [33-68,L62W]
Synonyms:
AMPL_PIG | Cytosol aminopeptidase | LAP3 | Leucine aminopeptidase (LAP)
Type:
Enzyme
Mol. Mass.:
4015.44
Organism:
Sus scrofa (Pig)
Description:
P28839[33-68,L62W]
Residue:
36
Sequence:
TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
  
Inhibitor
Name:
BDBM50025099
Synonyms:
CHEMBL3355111
Type:
Small organic molecule
Emp. Form.:
C19H26N3O4P
Mol. Mass.:
391.4012
SMILES:
NCc1cccc(CC(CP(O)(=O)C(N)CCc2ccncc2)C(O)=O)c1
Structure:
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