Reaction Details Report a problem with these data
Target
Adiponectin receptor protein 2
Ligand
BDBM50059083
Substrate
n/a
Meas. Tech.
ChEMBL_1461018 (CHEMBL3395076)
Kd
3100±n/a nM
Citation
 Rana, S; Blowers, EC; Natarajan, A Small molecule adenosine 5'-monophosphate activated protein kinase (AMPK) modulators and human diseases. J Med Chem 58:2-29 (2015) [PubMed]  Article 
Target
Name:
Adiponectin receptor protein 2
Synonyms:
ADIPOR2 | Adiponectin receptor protein 2 | PAQR2 | PAQR2_HUMAN | Progestin and adipoQ receptor family member II
Type:
PROTEIN
Mol. Mass.:
43884.36
Organism:
Homo sapiens (Human)
Description:
ChEMBL_109559
Residue:
386
Sequence:
MNEPTENRLGCSRTPEPDIRLRKGHQLDGTRRGDNDSHQGDLEPILEASVLSSHHKKSSEEHEYSDEAPQEDEGFMGMSPLLQAHHAMEKMEEFVCKVWEGRWRVIPHDVLPDWLKDNDFLLHGHRPPMPSFRACFKSIFRIHTETGNIWTHLLGCVFFLCLGIFYMFRPNISFVAPLQEKVVFGLFFLGAILCLSFSWLFHTVYCHSEGVSRLFSKLDYSGIALLIMGSFVPWLYYSFYCNPQPCFIYLIVICVLGIAAIIVSQWDMFATPQYRGVRAGVFLGLGLSGIIPTLHYVISEGFLKAATIGQIGWLMLMASLYITGAALYAARIPERFFPGKCDIWFHSHQLFHIFVVAGAFVHFHGVSNLQEFRFMIGGGCSEEDAL
  
Inhibitor
Name:
BDBM50059083
Synonyms:
CHEMBL3393145
Type:
Small organic molecule
Emp. Form.:
C27H28N2O3
Mol. Mass.:
428.5228
SMILES:
O=C(COc1ccc(cc1)C(=O)c1ccccc1)NC1CCN(Cc2ccccc2)CC1
Structure:
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