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Target
RAF proto-oncogene serine/threonine-protein kinase
Ligand
BDBM50172058
Substrate
n/a
Meas. Tech.
ChEMBL_1577193 (CHEMBL3807567)
IC50
22800±n/a nM
Citation
More Info.:
Target
Name:
RAF proto-oncogene serine/threonine-protein kinase
Synonyms:
Craf | Proto-oncogene c-RAF | RAF proto-oncogene serine/threonine-protein kinase | RAF1_MOUSE | Raf-1 | Raf1
Type:
PROTEIN
Mol. Mass.:
72947.25
Organism:
Mus musculus
Description:
ChEMBL_116790
Residue:
648
Sequence:
MEHIQGAWKTISNGFGLKDAVFDGSSCISPTIVQQFGYQRRASDDGKLTDSSKTSNTIRVFLPNKQRTVVNVRNGMSLHDCLMKALKVRGLQPECCAVFRLLQEHKGKKARLDWNTDAASLIGEELQVDFLDHVPLTTHNFARKTFLKLAFCDICQKFLLNGFRCQTCGYKFHEHCSTKVPTMCVDWSNIRQLLLFPNSTVGDSGVPAPPSFPMRRMRESVSRMPASSQHRYSTPHAFTFNTSSPSSEGSLSQRQRSTSTPNVHMVSTTLHVDSRMIEDAIRSHSESASPSALSSSPNNLSPTGWSQPKTPVPAQRERAPGSGTQEKNKIRPRGQRDSSYYWEIEASEVMLSTRIGSGSFGTVYKGKWHGDVAVKILKVVDPTPEQLQAFRNEVAVLRKTRHVNILLFMGYMTKDNLAIVTQWCEGSSLYKHLHVQETKFQMFQLIDIARQTAQGMDYLHAKNIIHRDMKSNNIFLHEGLTVKIGDFGLATVKSRWSGSQQVEQPTGSVLWMAPEVIRMQDDNPFSFQSDVYSYGIVLYELMAGELPYAHINNRDQIIFMVGRGYASPDLSRLYKNCPKAMKRLVADCVKKVKEERPLFPQILSSIELLQHSLPKINRSASEPSLHRAAHTEDINACTLTTSPRLPVF