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Target
Polyprotein II
Ligand
BDBM50212470
Substrate
n/a
Meas. Tech.
ChEBML_28873
IC50
>1110000±n/a nM
Citation
  TBA Bioorg Med Chem Lett 2:145-148 (1992)   
Target
Name:
Polyprotein II
Synonyms:
Avian myoblastosis virus polyprotein II
Type:
PROTEIN
Mol. Mass.:
98728.91
Organism:
Avian myeloblastosis virus
Description:
ChEMBL_331788
Residue:
893
Sequence:
IGRATVLTVALHLAIPLKWKPNHTPVWIDQWPLPEGKLVALTQLVEKELQLGHIEPSLSCWNTPVFVIRKASGSYRLLHDLRAVNAKLVPFGAVQQGAPVLSALPRGWPLMVLDLKDCFFSIPLAEQDREAFAFTLPSVNNQAPARRFQWKVLPQGMTCSPTICQLIVGQILEPLRLKHPSLRMLHYMDDLLLAASSHDGLEAAGEEVISTLERAGFTISPDKVQREPGVQYLGYKLGSTYVAPVGLVAEPRIATLWDVQKLVGSLQWLRPALGIPPRLRGPFYEQLRGSDPNEAREWNLDMKMAWREIVRLSTTAALERWDPALPLEGAVARCEQGAIGVLGQGLSTHPRPCLWLFSTQPTKAFTAWLEVLTLLITKLRASAVRTFGKEVDILLLPACFRDDLPLPEGILLALRGFAGKIRSSDTPSIFDIARPLHVSLKVRVTDHPVPGPTVFTDASSSTHKGVVVWREGPRWEIKEIADLGASVQQLEARAVAMALLLWPTTPTNVVTDSAFVAKMLLKMGQEGVPSTAAAFILEDALSQRSAMAAVLHVRSHSEVPGFFTEGNDVADSQATFQAYPLREAKDLHTALHIGPRALSKACNISMQQAREVVQTCPHCNSAPALEAGVNPRGLGPLQIWQTDFTLEPRMAPRSWLAVTVDTASSAIVVTQHGRVTSVAAQHHWATAIAVLGRPKAIKTDNGSCFTSKSTREWLARWGIAHTTGIPGNSQGQAMVERANRLLKDKIRVLAEGDGFMKRIPTSKQGELLAKAMYALNHFERGENTKTPIQKHWRPTVLTEGPPVKIRIETGEWEKGWNVLVWGRGYAAVKNRDTDKVIWVPSRKVKPDIAQKDEVTKKDEASPLFAGWRHIDKRIITLHSSFSKINLLVCFIFH
  
Inhibitor
Name:
BDBM50212470
Synonyms:
CHEMBL605695
Type:
Small organic molecule
Emp. Form.:
C10H13F2N2O8P
Mol. Mass.:
358.1894
SMILES:
O[C@@H]1[C@@H](COP(O)(=O)C(F)F)OC([C@@H]1O)n1ccc(=O)[nH]c1=O |r|
Structure:
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