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TargetBeta-2 adrenergic receptor and beta-3 adrenergic receptor
LigandBDBM50232757
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1648545
Kd 0.018197±n/a nM
Citation Schmidt, DGunera, JBaker, JGKolb, P Similarity- and Substructure-Based Development of฿ ACS Med Chem Lett8:481-485 (2017) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Beta-2 adrenergic receptor and beta-3 adrenergic receptor
Name:Beta-2 adrenergic receptor and beta-3 adrenergic receptor
Synonyms:ADRB2 | ADRB2R | B2AR | Beta-2 adrenergic receptor | Beta-2 adrenoceptor | Beta-2 adrenoreceptor
Type:n/a
Mol. Mass.:46461.69
Organism:Homo sapiens (Human)
Description:P07550
Residue:413
Sequence:
MGQPGNGSAFLLAPNGSHAPDHDVTQERDEVWVVGMGIVMSLIVLAIVFGNVLVITAIAK
FERLQTVTNYFITSLACADLVMGLAVVPFGAAHILMKMWTFGNFWCEFWTSIDVLCVTAS
IETLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQE
AINCYANETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKRQLQKIDKSEGRF
HVQNLSQVEQDGRTGHGLRRSSKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQD
NLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCLRRSSLKAYGNGYSSNGNT
GEQSGYHVEQEKENKLLCEDLPGTEDFVGHQGTVPSDNIDSQGRNCSTNDSLL
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  Blast E-value cutoff:
BDBM50232757
NameBDBM50232757
Synonyms:CHEMBL4092412
TypeSmall organic molecule
Emp. Form.C19H25NO2
Mol. Mass.299.4073
SMILESCC(C)(C)NC[C@@H](O)COc1ccccc1-c1ccccc1 |r|
Structure
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n/a