Target
Neuropeptide Y receptor type 2
Ligand
BDBM50015490
Substrate
n/a
Ki
1.8±n/a nM
Comments
PDSP_1370
Citation
 Weinberg, DHSirinathsinghji, DJTan, CPShiao, LLMorin, NRigby, MRHeavens, RHRapoport, DRBayne, MLCascieri, MAStrader, CDLinemeyer, DLMacNeil, DJ Cloning and expression of a novel neuropeptide Y receptor. J Biol Chem 271:16435-8 (1996) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 2
Synonyms:
NPY-Y2 | NPY2R_MOUSE | Npy2r | Npy2r protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42634.12
Organism:
MOUSE
Description:
P97295
Residue:
381
Sequence:
MGPVGAEADENQTVEVKVEPYGPGHTTPRGELPPDPEPELIDSTKLVEVQVILILAYCSIILLGVVGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGPVLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLASPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSVYGTVYSLSTLLILYVLPLGIISFSYTRIWSKLRNHVSPGAASDHYHQRRHKMTKMLVCVVVVFAVSWLPLHAFQLAVDIDSHVLDLKEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSMTFKAKKNLEVKKNNGPTDSFSEATNV
  
Inhibitor
Name:
BDBM50015490
Synonyms:
CHEMBL438945 | H-YPSKPDNPGEDAPAEDMARYYSALRHYINLITRQRY-NH2 | NPY | NPY, human | NPY, human, rat | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly-Glu-Asp-Ala-Pro- Ala-Glu-Asp-Met-Ala-Arg-Tyr-Tyr-Ser-Ala-Leu-Arg-His- Tyr-Ile-Asn-Leu-Ile-Thr-Arg-Gln-Arg-Tyr-NH2 (NPY) | human Neuropeptide Y
Type:
Small organic molecule
Emp. Form.:
C189H285N55O57S
Mol. Mass.:
4271.685
SMILES:
n/a
Structure:
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