Reaction Details
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5-hydroxytryptamine receptor 1D
Ligand
BDBM82272
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_7268
Citation
Baxter, GS Novel discriminatory ligands for 5-HT2B receptors. Behav Brain Res 73:149-52 (1996) [PubMed] Article More Info.:
Target
Name:
5-hydroxytryptamine receptor 1D
Synonyms:
5-HT1D | 5-hydroxytryptamine receptor 1D | 5HT1D_CAVPO | HTR1D | Serotonin 1d (5-HT1d) receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
41780.38
Organism:
GUINEA PIG
Description:
5-HT1D HTR1D GUINEA PIG::Q60484
Residue:
376
Sequence:
MSPPNQSEEGLPQEASNRSLNATETPGDWDPGLLQALKVSLVVVLSIITLATVLSNAFVLTTILLTRKLHTPANYLIGSLATTDLLVSILVMPISIAYTTTRTWNFGQILCDIWVSSDITCCTASILHLCVIALDRYWAITDALEYSKRRTAGHAGAMIAAVWVISICISIPPLFWRQAQAQEEMSDCLVNTSQISYTIYSTCGAFYIPSVLLIILYSRIYRAARSRILNPPSLSGKRFTTAHLITGSAGSSLCSLNPSLHEGHMHPGSPLFFNHVRIKLADSVLERKRISAARERKATKTLGIILGAFIVCWLPFFVVSLVLPICRDSCWIHPALFDFFTWLGYLNSLINPIIYTVFNEDFRQAFQKVVHFRKAS
Inhibitor
Name:
BDBM82272
Synonyms:
SB 200646 | SB200646a
Type:
n/a
Emp. Form.:
C15H14N4O
Mol. Mass.:
266.2979
SMILES:
Cn1ccc2cc(NC(=O)Nc3cccnc3)ccc12
Structure:
