Reaction Details Report a problem with these data
Target
5-hydroxytryptamine receptor 4
Ligand
BDBM82087
Substrate
n/a
Ki
524.8±n/a nM
Comments
PDSP_172
Citation
 Claeysen, S; Sebben, M; Journot, L; Bockaert, J; Dumuis, A Cloning, expression and pharmacology of the mouse 5-HT(4L) receptor. FEBS Lett 398:19-25 (1996) [PubMed]  Article 
Target
Name:
5-hydroxytryptamine receptor 4
Synonyms:
5-HT-4 | 5-HT4 | 5-HT4L | 5-hydroxytryptamine receptor 4 | 5HT4R_MOUSE | Htr4 | Serotonin 4 (5-HT4) receptor | Serotonin receptor 4
Type:
Enzyme Catalytic Domain
Mol. Mass.:
43970.99
Organism:
MOUSE
Description:
5-HT4 HTR4 MOUSE::P97288
Residue:
388
Sequence:
MDKLDANVSSNEGFRSVEKVVLLTFLAVVILMAILGNLLVMVAVCRDRQLRKIKTNYFIVSLAFADLLVSVLVMPFGAIELVQDIWAYGEMFCLVRTSLDVLLTTASIFHLCCISLDRYYAICCQPLVYRNKMTPLRIALMLGGCWVLPMFISFLPIMQGWNNIGIVDVIEKRKFSHNSNSTWCVFMVNKPYAITCSVVAFYIPFLLMVLAYYRIYVTAKEHAQQIQMLQRAGATSESRPQPADQHSTHRMRTETKAAKTLCVIMGCFCFCWAPFFVTNIVDPFIDYTVPEQVWTAFLWLGYINSGLNPFLYAFLNKSFRRAFLIILCCDDERYKRPPILGQTVPCSTTTINGSTHVLRDTVECGGQWESRCHLTATSPLVAAQPSDT
  
Inhibitor
Name:
BDBM82087
Synonyms:
2-(5-methoxy-1H-indol-3-yl)ethanamine | 5-MT | 5-Methoxytryptamine hydrochloride | CAS_66-83-1 | tryptamine, 5-Methoxy
Type:
Small organic molecule
Emp. Form.:
C11H14N2O
Mol. Mass.:
190.2417
SMILES:
COc1ccc2[nH]cc(CCN)c2c1
Structure:
Search PDB for entries with ligand similarity: