Reaction Details Report a problem with these data
Target
5-hydroxytryptamine receptor 1D
Ligand
BDBM85097
Substrate
n/a
Ki
398.1±n/a nM
Comments
PDSP_1670
Citation
Kennett, GA; Wood, MD; Bright, F; Trail, B; Riley, G; Holland, V; Avenell, KY; Stean, T; Upton, N; Bromidge, S; Forbes, IT; Brown, AM; Middlemiss, DN; Blackburn, TP SB 242084, a selective and brain penetrant 5-HT2C receptor antagonist. Neuropharmacology 36:609-20 (1997) [PubMed] Article
More Info.:
Target
Name:
5-hydroxytryptamine receptor 1D
Synonyms:
5-HT1D | HTR1D
Type:
Enzyme Catalytic Domain
Mol. Mass.:
41501.69
Organism:
C.H.O.
Description:
5-HT1D HTR1D C.H.O.::A0A1U8CB25
Residue:
374
Sequence:
MSLPNQSIEGLSQEASNRSLNTTGAWDPQILQALKISLVVVLSIITLATVLSNAFVLTTILLTKKLHTPANYLIGSLATTDLLVSILVMPISIAYTTTRTWNFGQILCDIWVSSDITCCTASILHLCVIALDRYWAITDALEYSKRRTAGHAAAMIAAVWAISICISIPPLFWRQATAHEEMSDCLVNTSQISYTIYSTCGAFYIPSILLIILYGRIYVAARSRILNPPSLYGKRFTTAQLITGSAGSSLCSLDPSLHDSHSHTVGSPLFFNQVKIKLADSILERKRISAARERKATKTLGIILGAFIICWLPFFVVSLVLPICRDSCWIHPALFDFFTWLGYLNSLINPVIYTVFNEDFRQAFQKVVHFRKAS