Ki Summary

Reaction Details

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Target

Galanin receptor type 3

Ligand

BDBM85170

Substrate

n/a

1000±n/a nM

Comments

PDSP_862

Citation

Borowsky, B; Walker, MW; Huang, LY; Jones, KA; Smith, KE; Bard, J; Branchek, TA; Gerald, C Cloning and characterization of the human galanin GALR2 receptor. Peptides 19:1771-81 (1998) [PubMed] Article

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Target

Name:

Galanin receptor type 3

Synonyms:

Type:

Enzyme Catalytic Domain

Mol. Mass.:

39599.97

Organism:

Homo sapiens (Human)

Description:

Galanin R3 GALR3 HUMAN::O60755

Residue:

368

Sequence:

MADAQNISLDSPGSVGAVAVPVVFALIFLLGTVGNGLVLAVLLQPGPSAWQEPGSTTDLFILNLAVADLCFILCCVPFQATIYTLDAWLFGALVCKAVHLLIYLTMYASSFTLAAVSVDRYLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDARRRALDVATFAAGYLLPVAVVSLAYGRTLRFLWAAVGPAGAAAAEARRRATGRAGRAMLAVAALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYALASRHFRARFRRLWPCGRRRRHRARRALRRVRPASSGPPGCPGDARPSGRLLAGGGQGPEPREGPVHGGEAARGPE

Inhibitor

Name:

BDBM85170

Synonyms:

Galanin (3-29), porcine

Type:

Small organic molecule

Emp. Form.:

C133H199N39O39

Mol. Mass.:

2968.2411

SMILES:

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Structure: