Target
Neuropeptide Y receptor type 1
Ligand
BDBM82421
Substrate
n/a
Ki
0.13±n/a nM
Comments
PDSP_1562
Citation
 Berglund, MMHolmberg, SKEriksson, HGedda, KMaffrand, JPSerradeil-Le Gal, CChhajlani, VGrundemar, LLarhammar, D The cloned guinea pig neuropeptide Y receptor Y1 conforms to other mammalian Y1 receptors. Peptides 20:1043-53 (1999) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 1
Synonyms:
FC5 | NPY-Y1 | NPY1-R | NPY1R_RAT | Neuropeptide Y receptor type 1 | Npy1r
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44126.41
Organism:
RAT
Description:
NPY-Y1 NPY1R RAT::P21555
Residue:
382
Sequence:
MNSTLFSRVENYSVHYNVSENSPFLAFENDDCHLPLAVIFTLALAYGAVIILGVSGNLALIIIILKQKEMRNVTNILIVNLSFSDLLVAVMCLPFTFVYTLMDHWVFGETMCKLNPFVQCVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYIGITVIWVLAVASSLPFVIYQILTDEPFQNVSLAAFKDKYVCFDKFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRRNNMMDKIRDSKYRSSETKRINVMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLLFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSKTSLKQASPVAFKKISMNDNEKI
  
Inhibitor
Name:
BDBM82421
Synonyms:
CAS_81858-94-8 | PYY, porcine
Type:
Small organic molecule
Emp. Form.:
C190H287N53O58
Mol. Mass.:
4241.6321
SMILES:
n/a
Structure:
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