Reaction Details
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Report a problem with these dataTarget
Adenosine receptor A3
Ligand
BDBM50053924
Substrate
n/a
Ki
3307±n/a nM
Comments
PDSP_2056
Citation
Durand, IH; Green, RD Cloning of a chick A3 adenosine receptor: characterization of ligand binding and receptor-effector coupling of chick A1 and A3 adenosine receptors. Naunyn Schmiedebergs Arch Pharmacol 363:81-6 (2001) [PubMed] Article More Info.:
Target
Name:
Adenosine receptor A3
Synonyms:
ADENOSINE A3 | ADORA3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
37723.59
Organism:
Chick
Description:
A0A8V1ACC1
Residue:
338
Sequence:
MCPQGSPCPASSSPINVTFNTSQVMGSIDVIYISAECLVALLAALGNIPVVWAVKLNAAFHNTTMYFIASLALADIAVGVFVVPLAVLVSLQVSIPFHFCLFLCCLMVVFTQASILSLLAIAIDRYLRVKLPIRYKIISTERRIWGALGLCWSLSLLVGLTPMFGWNKQRSAPYHTCGFTSVIRMDYMVYFSFFAWTLIPLSIMCALYVAVFYIIRTKLSQGATGARGAGTFYGKEFRKAKSLALILFLFAVSWLPLCIMNCVLYFHPEYKIPKPWIFLGILLSHANSAMNPVVYACKIKKFKTTYLLILRTYILCRKKPQAMPSSYRLNTPAVVDTE
Inhibitor
Name:
BDBM50053924
Synonyms:
3,6-Dichloro-2-(2-isopropoxy-4-methyl-phenyl)-chromen-4-one | CHEMBL89093 | MRS1067
Type:
Small organic molecule
Emp. Form.:
C19H16Cl2O3
Mol. Mass.:
363.235
SMILES:
CC(C)Oc1cc(C)ccc1-c1oc2ccc(Cl)cc2c(=O)c1Cl
Structure:
