Reaction Details Report a problem with these data
Target
Nicotinic acetylcholine receptor
Ligand
BDBM85224
Substrate
n/a
Ki
23±n/a nM
Comments
PDSP_1165
Citation
 Jensen, AA; Mikkelsen, I; Frølund, B; Bräuner-Osborne, H; Falch, E; Krogsgaard-Larsen, P Carbamoylcholine homologs: novel and potent agonists at neuronal nicotinic acetylcholine receptors. Mol Pharmacol 64:865-75 (2003) [PubMed]  Article 
Target
Name:
Nicotinic acetylcholine receptor
Synonyms:
Nicotinic acetylcholine receptor | n-AChR
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2478.99
Organism:
RAT
Description:
n-AChR 0 RAT::Q62594
Residue:
23
Sequence:
MTMALLGTLLLLALFGRSQGKNE
  
Inhibitor
Name:
BDBM85224
Synonyms:
CAS_1918-18-9 | MCC | SWEP
Type:
Small organic molecule
Emp. Form.:
C8H7Cl2NO2
Mol. Mass.:
220.053
SMILES:
COC(=O)Nc1ccc(Cl)c(Cl)c1
Structure:
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