Target
Trace amine-associated receptor 1
Ligand
BDBM109448
Substrate
n/a
Meas. Tech.
Radioligand Binding Assay
Ki
6.3±n/a nM
Citation
 Galley, GGroebke Zbinden, KNorcross, RStalder, H 2-aminooxazolines as TAAR1 ligands US Patent  US8604061 Publication Date 12/10/2013 
Target
Name:
Trace amine-associated receptor 1
Synonyms:
TAAR1_MOUSE | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1
Type:
Protein
Mol. Mass.:
37635.41
Organism:
Mus musculus (Mouse)
Description:
Q923Y8
Residue:
332
Sequence:
MHLCHAITNISHRNSDWSREVQASLYSLMSLIILATLVGNLIVIISISHFKQLHTPTNWLLHSMAIVDFLLGCLIMPCSMVRTVERCWYFGEILCKVHTSTDIMLSSASIFHLAFISIDRYCAVCDPLRYKAKINISTILVMILVSWSLPAVYAFGMIFLELNLKGVEELYRSQVSDLGGCSPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRTNVQVGLEGKSQAPQSKETKAAKTLGIMVGVFLVCWCPFFLCTVLDPFLGYVIPPSLNDALYWFGYLNSALNPMVYAFFYPWFRRALKMVLLGKIFQKDSSRSKLFL
  
Inhibitor
Name:
BDBM109448
Synonyms:
US8604061, 184
Type:
Small organic molecule
Emp. Form.:
C14H17F3N2O
Mol. Mass.:
286.2928
SMILES:
CCC(C[C@H]1COC(N)=N1)c1ccc(cc1)C(F)(F)F |r,c:8|
Structure:
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