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TargetTrypsin-1
LigandBDBM109660
Substrate/Competitorn/a
Meas. Tech.Inhibition Assay
Ki 0.23±0.0 nM
Citation Konishi, ATokumasu, MSuzuki, TKoshiba, TOhsumi, KIkehara, OKodama, Y Heteroarylcarboxylic acid ester derivative US Patent US8609715 Publication Date 12/17/2013
More Info.:Get all data from this article,  Assay Method
 
Trypsin-1
Name:Trypsin
Synonyms:Alpha-trypsin chain 1 | Alpha-trypsin chain 2 | Beta-trypsin | Cationic trypsinogen | Serine protease 1 | Trypsin
Type:Enzyme
Mol. Mass.:26557.80
Organism:Homo sapiens (human)
Description:P07477
Residue:247
Sequence:
MNPLLILTFVAAALAAPFDDDDKIVGGYNCEENSVPYQVSLNSGYHFCGGSLINEQWVVS
AGHCYKSRIQVRLGEHNIEVLEGNEQFINAAKIIRHPQYDRKTLNNDIMLIKLSSRAVIN
ARVSTISLPTAPPATGTKCLISGWGNTASSGADYPDELQCLDAPVLSQAKCEASYPGKIT
SNMFCVGFLEGGKDSCQGDSGGPVVCNGQLQGVVSWGDGCAQKNKPGVYTKVYNYVKWIK
NTIAANS
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  Blast E-value cutoff:
BDBM109660
n/a
NameBDBM109660
Synonyms:US8609715, A-68
TypeSmall organic molecule
Emp. Form.C23H19N3O8
Mol. Mass.465.4123
SMILESNC(=N)c1ccc(OC(=O)c2ccc(o2)-c2ccc(cc2)C(=O)N[C@@H](CC(O)=O)C(O)=O)cc1 |r|
Structure
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