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Reaction Details
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TargetTrace amine-associated receptor 1 (TAAR1)
LigandBDBM119204
Substrate/Competitorn/a
Meas. Tech.Radioligand Binding Assay
Ki 0.7±n/a nM
Citation Nettekoven, MNorcross, RPolara, A Dihydrooxazol-2-amine derivatives US Patent US8673950 Publication Date 3/18/2014
More Info.:Get all data from this article,  Assay Method
 
Trace amine-associated receptor 1 (TAAR1)
Name:Trace amine-associated receptor 1
Synonyms:Trace amine receptor 1 (TARR1) | Trace amine-associated receptor1
Type:Enzyme
Mol. Mass.:38034.73
Organism:Rattus norvegicus (Rat)
Description:Q923Y9
Residue:332
Sequence:
MHLCHNSANISHTNSNWSRDVRASLYSLISLIILTTLVGNLIVIISISHFKQLHTPTNWL
LHSMAVVDFLLGCLVMPYSMVRTVEHCWYFGELFCKLHTSTDIMLSSASILHLAFISIDR
YYAVCDPLRYKAKINLAAIFVMILISWSLPAVFAFGMIFLELNLEGVEELYHNQVFCLRG
CFPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRANLQVGLEGESRAPQ
SKETKAAKTLGIMVGVFLLCWCPFFFCMVLDPFLGYVIPPTLNDTLNWFGYLNSAFNPMV
YAFFYPWFRRALKMVLFGKIFQKDSSRSKLFL
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM119204
NameBDBM119204
Synonyms:US8673950, 72
TypeSmall organic molecule
Emp. Form.C16H18ClN5O
Mol. Mass.331.8
SMILESCc1cc(CC[C@H]2COC(N)=N2)ccc1Nc1ncc(Cl)cn1 |r,c:10|
Structure
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