Reaction Details Report a problem with these data
Target
Somatostatin receptor type 5
Ligand
BDBM123316
Substrate
n/a
Meas. Tech.
Binding Assay
pH
7.8±n/a
IC50
86.02±n/a nM
Comments
extracted
Citation
Duffy, JL; Bao, J; Ondeyka, DL; Tyagarajan, S; Shao, P; Ye, F; Katipally, R; Zwicker, A; Sherer, EC; Plotkin, MA; Moningka, R; Hussain, Z; Wood, HB; Ujjainwalla, F; Romero, FA; Finke, PE; Zang, Y; Liu, W Spiroxazolidinone compounds US Patent US8742110 Publication Date 6/3/2014
More Info.:
Target
Name:
Somatostatin receptor type 5
Synonyms:
SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5)
Type:
Enzyme
Mol. Mass.:
39218.02
Organism:
Homo sapiens (Human)
Description:
P35346
Residue:
364
Sequence:
MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTLVIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDGVNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADVQEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRRRSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCANPVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQTSKL