Reaction Details Report a problem with these data
Target
Trace amine-associated receptor 7b
Ligand
BDBM129526
Substrate
n/a
Meas. Tech.
Radioligand Binding
pH
7.4±n/a
Temperature
310.15±n/a K
Ki
6.5±n/a nM
Comments
extracted
Citation
Galley, G; Norcross, RD; Pflieger, P Heterocyclic amine derivatives US Patent US8802673 Publication Date 8/12/2014
More Info.:
Target
Name:
Trace amine-associated receptor 7b
Synonyms:
TAA7B_RAT | Ta12 | Taar7b | Tar12 | Trace amine-associated receptor 1 (TAAR1) | Trar12
Type:
Enzyme
Mol. Mass.:
40296.65
Organism:
Rattus norvegicus (Rat)
Description:
Q923X8
Residue:
358
Sequence:
MATDDDRFPWDQDSILSRDLLSASSMQLCYEKLNRSCVRSPYSPGPRLILYAVFGFGAVLAVCGNLLVMTSILHFRQLHSPANFLVASLACADFLVGLTVMPFSMVRSVEGCWYFGDIYCKFHSSFDGSFCYSSIFHLCFISADRYIAVSDPLIYPTRFTASVSGKCITFSWLLSIIYSFSLFYTGVNEAGLEDLVSALTCVGGCQIAVNQSWVFINFLLFLVPALVMMTVYSKIFLIAKQQAQNIEKMGKQTARASESYKDRVAKRERKAAKTLGIAVAAFLLSWLPYFIDSIIDAFLGFVTPTYVYEILVWIGYYNSAMNPLIYAFFYPWFRKAIKLIVTGKILRENSSATNLFPE