Reaction Details Report a problem with these data
Target
Protein mono-ADP-ribosyltransferase PARP15 [460-656]
Ligand
BDBM199181
Substrate
n/a
Meas. Tech.
Enzymatic Activity Assay
IC50
>1.0e+4±n/a nM
Citation
Venkannagari, H; Verheugd, P; Koivunen, J; Haikarainen, T; Obaji, E; Ashok, Y; Narwal, M; Pihlajaniemi, T; Lüscher, B; Lehtiö, L Small-Molecule Chemical Probe Rescues Cells from Mono-ADP-Ribosyltransferase ARTD10/PARP10-Induced Apoptosis and Sensitizes Cancer Cells to DNA Damage. Cell Chem Biol 23:1251-1260 (2016) [PubMed] Article
More Info.:
Target
Name:
Protein mono-ADP-ribosyltransferase PARP15 [460-656]
Synonyms:
BAL3 | Human diphtheria toxin-like ADP-ribosyltransferase (ARTD7 or PARP15) | PAR15_HUMAN | PARP15
Type:
n/a
Mol. Mass.:
22502.60
Organism:
Homo sapiens (Human)
Description:
Q460N3[460-656]
Residue:
197
Sequence:
MKKRDLSASLNFQSTFSMTTCNLPEHWTDMNHQLFCMVQLEPGQSEYNTIKDKFTRTCSSYAIEKIERIQNAFLWQSYQVKKRQMDIKNDHKNNERLLFHGTDADSVPYVNQHGFNRSCAGKNAVSYGKGTYFAVDASYSAKDTYSKPDSNGRKHMYVVRVLTGVFTKGRAGLVTPPPKNPHNPTDLFDSVTNNTRS