Reaction Details Report a problem with these data
Target
Protein mono-ADP-ribosyltransferase PARP14 [1535-1801]
Ligand
BDBM199181
Substrate
n/a
Meas. Tech.
Enzymatic Activity Assay
IC50
2.3e+4±n/a nM
Citation
Venkannagari, H; Verheugd, P; Koivunen, J; Haikarainen, T; Obaji, E; Ashok, Y; Narwal, M; Pihlajaniemi, T; Lüscher, B; Lehtiö, L Small-Molecule Chemical Probe Rescues Cells from Mono-ADP-Ribosyltransferase ARTD10/PARP10-Induced Apoptosis and Sensitizes Cancer Cells to DNA Damage. Cell Chem Biol 23:1251-1260 (2016) [PubMed] Article
More Info.:
Target
Name:
Protein mono-ADP-ribosyltransferase PARP14 [1535-1801]
Synonyms:
BAL2 | Human diphtheria toxin-like ADP-ribosyltransferase (ARTD8 or PARP14) | KIAA1268 | PAR14_HUMAN | PARP14
Type:
n/a
Mol. Mass.:
30839.62
Organism:
Homo sapiens (Human)
Description:
Q460N5[1535-1801]
Residue:
267
Sequence:
IEWQYNDNNTSHCFNKMTNLKLEDARREKKKTVDVKINHRHYTVNLNTYTATDTKGHSLSVQRLTKSKVDIPAHWSDMKQQNFCVVELLPSDPEYNTVASKFNQTCSHFRIEKIERIQNPDLWNSYQAKKKTMDAKNGQTMNEKQLFHGTDAGSVPHVNRNGFNRSYAGKNAVAYGKGTYFAVNANYSANDTYSRPDANGRKHVYYVRVLTGIYTHGNHSLIVPPSKNPQNPTDLYDTVTDNVHHPSLFVAFYDYQAYPEYLITFRK