Reaction Details | |||
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Target | Ephrin type-A receptor 2 (EPHA2) | ||
Ligand | BDBM209862 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | Kinobeads Competition Assay | ||
Kd | 265±0.0 nM | ||
Citation | ![]() | ||
More Info.: | Get all data from this article, Assay Method | ||
Ephrin type-A receptor 2 (EPHA2) | |||
Name: | Ephrin type-A receptor 2 (EPHA2) | ||
Synonyms: | n/a | ||
Type: | Protein | ||
Mol. Mass.: | 34367.96 | ||
Organism: | Homo sapiens (Human) | ||
Description: | EPHA2 truncation (596-900 aa); 519U | ||
Residue: | 305 | ||
Sequence: |
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BDBM209862 | |||
Name | BDBM209862 | ||
Synonyms: | 4-(3-chloro-2-fluorophenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acid | MK-5108 | ||
Type | Small organic molecule | ||
Emp. Form. | C22H21ClFN3O3S | ||
Mol. Mass. | 461.937 | ||
SMILES | OC(=O)C1(Cc2cccc(Nc3nccs3)n2)CCC(CC1)Oc1cccc(Cl)c1F |(6.1,3.85,;7.64,3.85,;8.41,5.18,;8.41,2.52,;9.18,3.85,;10.72,3.85,;11.49,5.18,;13.03,5.18,;13.8,3.85,;13.03,2.52,;13.8,1.18,;15.35,1.18,;16.25,-.06,;17.71,.41,;17.71,1.95,;16.25,2.43,;11.49,2.52,;7.08,1.75,;7.08,.21,;8.41,-.56,;9.75,.21,;9.75,1.75,;8.41,-2.1,;7.08,-2.87,;7.08,-4.41,;5.75,-5.18,;4.41,-4.41,;4.41,-2.87,;3.08,-2.1,;5.75,-2.1,;5.75,-.56,)| | ||
Structure | ![]() | ||
n/a |