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TargetCyclin-dependent kinase 2
LigandBDBM8068
Substrate/Competitorn/a
Meas. Tech.OctetRed_Method3
KOFF 5.62E-02 s-1
Citation D3R, DD CSAR CDK2 Kinase D3R D3R Publication Date 6/30/2015
More Info.:Get all data from this article,  Assay Method
 
Cyclin-dependent kinase 2
Name:Protein cereblon/Cyclin-dependent kinase 2
Synonyms:CDK2 | CDK2-Kinase | Cell division protein kinase 2 | Cyclin-dependent kinase 2 (CDK2) | p33 protein kinase
Type:Enzyme Subunit
Mol. Mass.:33938.17
Organism:Homo sapiens (Human)
Description:P24941
Residue:298
Sequence:
MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNH
PNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHS
HRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYTHEVVTLWYRAPEILLGCKYY
STAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSF
PKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL
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  Blast E-value cutoff:
BDBM8068
NameBDBM8068
Synonyms:2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 39 | 2-Chloro-N4-[4-(2,4-dimethylthiazol-5-yl)pyrimidin-2-yl]-N1,N1-dimethylbenzene-1,4-diamine | 2-chloro-4-N-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-1-N,1-N-dimethylbenzene-1,4-diamine | CS20
TypeSmall organic molecule
Emp. Form.C17H18ClN5S
Mol. Mass.359.876
SMILESCN(C)c1ccc(Nc2nccc(n2)-c2sc(C)nc2C)cc1Cl
Structure
n/a