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Target
Cholesteryl ester transfer protein
Ligand
BDBM234611
Substrate
n/a
Meas. Tech.
In Vitro Radioactive Assays of CETP-Catalyzed CE and TG Transfer (RTA Assay)
pH
7.4±n/a
Temperature
310.15±n/a K
IC50
3±n/a nM
Comments
extracted
Citation
Acton, III, JJ; Ye, F; Vachal, P; Sha, D; Dropinski, JF; Chu, L; Ondeyka, D; Kim, AJ; Colandrea, VJ; Zang, Y; Zhang, F; Dong, G Cyclic amine substituted heterocyclic CETP inhibitors US Patent US9353101 Publication Date 5/31/2016
More Info.:
Target
Name:
Cholesteryl ester transfer protein
Synonyms:
CETP | CETP_HUMAN | Cholesteryl ester transfer protein (CETP) | Lipid transfer protein I
Type:
Enzyme
Mol. Mass.:
54751.53
Organism:
Homo sapiens (Human)
Description:
P11597
Residue:
493
Sequence:
MLAATVLTLALLGNAHACSKGTSHEAGIVCRITKPALLVLNHETAKVIQTAFQRASYPDITGEKAMMLLGQVKYGLHNIQISHLSIASSQVELVEAKSIDVSIQNVSVVFKGTLKYGYTTAWWLGIDQSIDFEIDSAIDLQINTQLTCDSGRVRTDAPDCYLSFHKLLLHLQGEREPGWIKQLFTNFISFTLKLVLKGQICKEINVISNIMADFVQTRAASILSDGDIGVDISLTGDPVITASYLESHHKGHFIYKNVSEDLPLPTFSPTLLGDSRMLYFWFSERVFHSLAKVAFQDGRLMLSLMGDEFKAVLETWGFNTNQEIFQEVVGGFPSQAQVTVHCLKMPKISCQNKGVVVNSSVMVKFLFPRPDQQHSVAYTFEEDIVTTVQASYSKKKLFLSLLDFQITPKTVSNLTESSSESVQSFLQSMITAVGIPEVMSRLEVVFTALMNSKGVSLFDIINPEIITRDGFLLLQMDFGFPEHLLVDFLQSLS