Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 1C87
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Graduate University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50118744(2-(carboxyformamido)-5,7-dihydro-4H-thieno[2,3-c]p...)
Affinity DataKi:  1.39E+4nMAssay Description:Binding affinity to PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Graduate University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50118744(2-(carboxyformamido)-5,7-dihydro-4H-thieno[2,3-c]p...)
Affinity DataKi:  1.40E+4nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Graduate University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50118744(2-(carboxyformamido)-5,7-dihydro-4H-thieno[2,3-c]p...)
Affinity DataKi:  1.41E+4nMAssay Description:Binding affinity to human recombinant PTP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)