Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) for PDB: 1JG0
TargetThymidylate synthase(Escherichia coli)
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LigandPNGBDBM50161779((S)-2-(5-Dimethylamino-naphthalene-1-sulfonylamino...)
Affinity DataKi:  1.80E+3nMAssay Description:All compounds were screened for inhibitory activity against Lactobacillus casei thymidylate synthase (LcTS) and Escherichia coli thymidylate synthase...More data for this Ligand-Target Pair
TargetThymidylate synthase(Escherichia coli)
Università

Curated by ChEMBL
LigandPNGBDBM50161779((S)-2-(5-Dimethylamino-naphthalene-1-sulfonylamino...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibitory constant against thymidylate synthase from Escherichia coliMore data for this Ligand-Target Pair
TargetThymidylate synthase(Escherichia coli)
Università

LigandPNGBDBM50161779((S)-2-(5-Dimethylamino-naphthalene-1-sulfonylamino...)
Affinity DataIC50:  5.00E+3nMAssay Description:Affinity assay of specificities of thymidylate synthase (TS)inhibitorsMore data for this Ligand-Target Pair