Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) for PDB: 1RT2
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50050533(TNK-651 | 6-BENZYL-1-BENZYLOXYMETHYL-5-ISOPROPYL U...)
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetReverse transcriptase(Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050533(TNK-651 | 6-BENZYL-1-BENZYLOXYMETHYL-5-ISOPROPYL U...)
Affinity DataIC50: 16nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetReverse transcriptase(Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050533(TNK-651 | 6-BENZYL-1-BENZYLOXYMETHYL-5-ISOPROPYL U...)
Affinity DataIC50: 20nMAssay Description:Inhibition of HIV1 reverse transcriptase using poly(ra)/oligo(dT)15 homopolymer template as substrate after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetReverse transcriptase(Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050533(TNK-651 | 6-BENZYL-1-BENZYLOXYMETHYL-5-ISOPROPYL U...)
Affinity DataIC50: 40nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetReverse transcriptase(Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050533(TNK-651 | 6-BENZYL-1-BENZYLOXYMETHYL-5-ISOPROPYL U...)
Affinity DataIC50: 88nMAssay Description:Inhibition of HIV1 reverse transcriptase after 1 hr by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)