Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 2BUA
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM11555((1-phenylcyclopentyl)methanamine | CHEMBL382127 | ...)
Affinity DataIC50: 3.00E+4nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
Santhera Pharmaceuticals

LigandPNGBDBM11555((1-phenylcyclopentyl)methanamine | CHEMBL382127 | ...)
Affinity DataIC50: 3.30E+4nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
Santhera Pharmaceuticals

LigandPNGBDBM11555((1-phenylcyclopentyl)methanamine | CHEMBL382127 | ...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
Santhera Pharmaceuticals

LigandPNGBDBM11555((1-phenylcyclopentyl)methanamine | CHEMBL382127 | ...)
Affinity DataIC50: 4.00E+4nMAssay Description:Binding affinity to DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)