Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) for PDB: 2POB
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423010(CHEMBL230259)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayChecked by AuthorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423010(CHEMBL230259)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of BRL-49653 stimulated human PPARgamma transactivation in CV-1 cells by GAL4 reporter assayChecked by AuthorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423010(CHEMBL230259)
Affinity DataEC50:  1.00E+3nMAssay Description:Transactivation of human PPARgamma in CV-1 cells by GAL4 reporter assayChecked by AuthorMore data for this Ligand-Target Pair