Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) for PDB: 2VWX
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM25223(2,4-Pyrimidine derivative, 25 | 3-({4-[(5-chloro-2...)
Affinity DataIC50:  40nMpH: 7.4 T: 2°CAssay Description:This assay detects inhibitors of EphB4-mediated phosphorylation of a polypeptide substrate using Alphascreen luminescence detection technology. The r...More data for this Ligand-Target Pair
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM25223(2,4-Pyrimidine derivative, 25 | 3-({4-[(5-chloro-2...)
Affinity DataIC50:  40nMAssay Description:Inhibition of EphB4More data for this Ligand-Target Pair
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM25223(2,4-Pyrimidine derivative, 25 | 3-({4-[(5-chloro-2...)
Affinity DataIC50:  172nMAssay Description:Inhibition of Myc-His-tagged EphB4 expressed in CHOK1 cells assessed as phosphorylation by ELISAMore data for this Ligand-Target Pair