Report error Found 14 Enz. Inhib. hit(s) for PDB: 2Y6O
Affinity DataKd: 0.0900nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKd: 0.0930nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.0930nMAssay Description:Binding constant for EPHA3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.240nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.240nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 0.240nMAssay Description:Binding constant for EPHA5 kinase domainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Nano Luc-fused full length C-terminal EPHA3 (unknown origin) expressed in HEK293T cells using NanoGlo as substrate incubated for 2 hrs ...More data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of Nano Luc-fused full length C-terminal EPHA5 (unknown origin) expressed in HEK293T cells using NanoGlo as substrate incubated for 2 hrs ...More data for this Ligand-Target Pair
Affinity DataKd: 3.70nMAssay Description:Binding affinity to human EPHA5 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibition of Nano Luc-fused full length C-terminal EPHA4 (unknown origin) expressed in HEK293T cells using NanoGlo as substrate incubated for 2 hrs ...More data for this Ligand-Target Pair
Affinity DataKd: 7.30nMAssay Description:Binding affinity to human EPHA4 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair