Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 3OMQ
TargetEstrogen receptor beta(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50341433(2-(trifluoromethylsulfonyl)-1,2,3,4-tetrahydroisoq...)
Affinity DataEC50:  310nMAssay Description:Transcriptional activation of human ERbeta receptor transfected in human U2OS cells assessed as increase of luciferase activity by estrogen response ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor beta(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50341433(2-(trifluoromethylsulfonyl)-1,2,3,4-tetrahydroisoq...)
Affinity DataEC50:  600nMAssay Description:Agonist activity at human N-terminal His6-tagged ERbeta receptor LBD expressed in Escherichia coli BL21 (DE3) assessed as induction of SRC1 peptide r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)