Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 3VW6
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Pharmadesign

Curated by ChEMBL
LigandPNGBDBM50334268(CHEMBL2205637 | CHEMBL1642655 | N-(6-(1H-imidazol-...)
Affinity DataIC50: 14nMAssay Description:Inhibition of ASK1 assessed as phosphorylated fluorescent peptide by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Pharmadesign

Curated by ChEMBL
LigandPNGBDBM50334268(CHEMBL2205637 | CHEMBL1642655 | N-(6-(1H-imidazol-...)
Affinity DataIC50: 14nMAssay Description:Competitive inhibition of human recombinant N-terminal FLAG-tagged ASK1 expressed in baculovirus infected Sf2 cells after 60 mins by scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)